Co-reporter:Ziqiang Liu;Lei Chen;Jing Li;Ke Liu;Jiaqi Zhao;Mengmeng Xu;Ren-zhong Wan;Wei Li;Lei Liu
Organic & Biomolecular Chemistry 2017 vol. 15(Issue 36) pp:7600-7606
Publication Date(Web):2017/09/20
DOI:10.1039/C7OB01793F
A modular and efficient method for the synthesis of α-substituted 1,2-dihydroquinolines is described. Under mild metal-free conditions, readily available N-carbamoyl 1,2-dihydroquinolines undergo oxidative C–H alkynylation, alkenylation, and allylation with a range of potassium trifluoroborates using TEMPO oxoammonium salt as an oxidant.
Co-reporter:Ziqiang Liu;Lei Chen;Jing Li;Ke Liu;Jiaqi Zhao;Mengmeng Xu;Ren-zhong Wan;Wei Li;Lei Liu
Organic & Biomolecular Chemistry 2017 vol. 15(Issue 36) pp:7600-7606
Publication Date(Web):2017/09/20
DOI:10.1039/C7OB01793F
A modular and efficient method for the synthesis of α-substituted 1,2-dihydroquinolines is described. Under mild metal-free conditions, readily available N-carbamoyl 1,2-dihydroquinolines undergo oxidative C–H alkynylation, alkenylation, and allylation with a range of potassium trifluoroborates using TEMPO oxoammonium salt as an oxidant.
Co-reporter:Aiping Huang, Lei Feng, Zhi Qiao, Wei Yu, Qingqing Zheng, Chen Ma
Tetrahedron 2013 69(2) pp: 642-646
Publication Date(Web):
DOI:10.1016/j.tet.2012.11.009